发明名称 PHARMACEUTICAL COMPOUNDS
摘要 The invention provides novel cryptophycin compounds which can be useful for disrupting the microtubulin system, as anti-neoplastic agents, and for the treatment of cancer. The invention further provides a formulation for administering the novel cryptophycin compounds.
申请公布号 WO9808505(A8) 申请公布日期 1999.08.12
申请号 WO1997US15240 申请日期 1997.08.29
申请人 ELI LILLY AND COMPANY;UNIVERSITY OF HAWAII;WAYNE STATE UNIVERSITY;AL-AWAR, RIMA, S.;EHLHARDT, WILLIAM, J.;GOTTUMUKKALA, SUBBARAJU, V.;MARTINELLI, MICHAEL, J.;MOHER, ERIC, D.;MOORE, RICHARD, E.;MUNROE, JOHN, E.;NORMAN, BRYAN, H.;PATEL, VINOD, F.;SHIH, CHUAN;TOTH, JOHN, E.;VASUDEVAN, VENKATRAGHAVAN;RAY, JAMES, E. 发明人 AL-AWAR, RIMA, S.;EHLHARDT, WILLIAM, J.;GOTTUMUKKALA, SUBBARAJU, V.;MARTINELLI, MICHAEL, J.;MOHER, ERIC, D.;MOORE, RICHARD, E.;MUNROE, JOHN, E.;NORMAN, BRYAN, H.;PATEL, VINOD, F.;SHIH, CHUAN;TOTH, JOHN, E.;VASUDEVAN, VENKATRAGHAVAN;RAY, JAMES, E.
分类号 A61K31/395;A61K31/427;A61K31/4427;A61K31/496;A61K31/7052;A61P35/00;A61P43/00;C07D273/00;C07D273/08;C07D281/00;C07D291/02;C07D413/06;C07D413/10;C07D413/12;C07D417/06;C07D417/14;C07F9/12;C07F9/6527;C07H15/26 主分类号 A61K31/395
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