发明名称 Spiro-azacyclic derivatives and their use as therapeutic agents
摘要 The present invention is directed to substituted spiro-azacyclic derivatives of the formula (I):(wherein R1, R2, R3, R4, R5, R6, R9, R10, X, Y, p and q are defined herein) which are tachykinin antagonists and are useful, for example, in the treatment or prevention of pain, inflammation, migraine, emesis and postherpetic neuralgia.
申请公布号 AU7067298(A) 申请公布日期 1998.11.24
申请号 AU19980070672 申请日期 1998.04.22
申请人 MERCK SHARP & DOHME LIMITED 发明人 NEIL ROY CURTIS;JASON MATTHEW ELLIOTT;GREGORY JOHN HOLLINGWORTH;PHILIPS STEPHEN JACKSON;JANUSZ JOZEF KULAGOWSKI;EILEEN MARY SEWARD;CHRISTOPHER JOHN SWAIN;BRIAN JOHN WILLIAMS
分类号 A61P25/04;A61K31/4192;A61K31/4196;A61K31/427;A61K31/433;A61K31/438;A61K31/4427;A61K31/497;A61K31/501;A61K31/506;A61K31/53;A61P1/08;A61P25/06;A61P29/00;A61P43/00;C07D491/10;C07D491/107 主分类号 A61P25/04
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