发明名称 ERYTHROMYCIN A DERIVATIVES
摘要 <p>Erythromycin A derivatives represented by general formula (I) or pharmaceutically acceptable salts thereof, each having a potent antibacterial activity against not only conventional erythromycin-sensitive bacteria but also erythromycin-resistant bacteria, wherein R?1 and R2¿ represent each group (a), group (b), pyridylacetyl, C¿4?-C8 cycloalkylmethyl, 1,2-bis(ethoxycarbonyl)vinyl, etc.; and A represents a group represented by -OC(=O)-R?17¿, -OC(=O)-CH¿2R?17, -OC(=O)-NH-R?17, -O-R17¿ or -OC(=O)-O-R17.</p>
申请公布号 WO1998023628(P1) 申请公布日期 1998.06.04
申请号 JP1997003687 申请日期 1997.10.14
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