| 发明名称 |
Muscarine antagonists |
| 摘要 |
This invention is concerned with novel 1,3-dihydro-1-[1-(1-heteroarylpiperidin-4-yl)piperidin-4-yl]-2H-benzimidazolones, derivatives thereof, their preparation, method of use and pharmaceutical compositions. These compounds are endowed with antimuscarinic activity and are useful in the treatment and/or prevention of myopia (commonly known as nearsightedness).
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| 申请公布号 |
US5756508(A) |
申请公布日期 |
1998.05.26 |
| 申请号 |
US19960736704 |
申请日期 |
1996.10.28 |
| 申请人 |
MERCK & CO., INC. |
发明人 |
THOMPSON, WAYNE J.;RANSOM, RICHARD W.;MALLORGA, PIERRE;SUGRUE, MICHAEL F. |
| 分类号 |
C07D401/14;C07D451/04;(IPC1-7):C07D211/14;C07D235/26;C07D239/26;A61K31/415 |
主分类号 |
C07D401/14 |
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