发明名称 |
1-AZONIABICYCLO[2.2.1]HEPTANE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
摘要 |
A compound of formula (I), wherein A is a divalent radical selected from A1)-O-CO-; A2)-CH2-O-CO; A3)-O-CH2-CO-; A4)-O-CH2-CH2-; A5)-N(R1)-CO-; A6)-N(R1)-CO-CO; A7)-N(R1)-CH2-CH2-; A8)-O-CH2-; wherein R1 is hydrogen or (C1-C4)alkyl, and Am is (1). Said compound is useful as a neurokinin receptor antagonist.
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申请公布号 |
WO9804561(A1) |
申请公布日期 |
1998.02.05 |
申请号 |
WO1997FR01393 |
申请日期 |
1997.07.25 |
申请人 |
SANOFI |
发明人 |
EMONDS-ALT, XAVIER;GUEULE, PATRICK;PROIETTO, VINCENZO;TAILLADES, JOELLE;VAN BROECK, DIDIER |
分类号 |
A61K31/4178;A61K31/422;A61K31/496;A61K31/5355;A61K31/5377;A61P43/00;C07D487/08;(IPC1-7):C07D487/08;A61K31/42;A61K31/535 |
主分类号 |
A61K31/4178 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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