发明名称 1-AZONIABICYCLO[2.2.1]HEPTANE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
摘要 A compound of formula (I), wherein A is a divalent radical selected from A1)-O-CO-; A2)-CH2-O-CO; A3)-O-CH2-CO-; A4)-O-CH2-CH2-; A5)-N(R1)-CO-; A6)-N(R1)-CO-CO; A7)-N(R1)-CH2-CH2-; A8)-O-CH2-; wherein R1 is hydrogen or (C1-C4)alkyl, and Am is (1). Said compound is useful as a neurokinin receptor antagonist.
申请公布号 WO9804561(A1) 申请公布日期 1998.02.05
申请号 WO1997FR01393 申请日期 1997.07.25
申请人 SANOFI 发明人 EMONDS-ALT, XAVIER;GUEULE, PATRICK;PROIETTO, VINCENZO;TAILLADES, JOELLE;VAN BROECK, DIDIER
分类号 A61K31/4178;A61K31/422;A61K31/496;A61K31/5355;A61K31/5377;A61P43/00;C07D487/08;(IPC1-7):C07D487/08;A61K31/42;A61K31/535 主分类号 A61K31/4178
代理机构 代理人
主权项
地址