摘要 |
<p>15-deoxy-spergualin analogues of formula (I) and their addn. salts are new. X = (CH2)n; Y = (CH2)4; T = (CH2)2; A = a single bond, -CH2-, -CH2O-, -CH2NH-, -CH(OH)-, -CHF-, or -CH(OCH3)-; n = 6-8. Intermediate cpds. of formula (II) are also claimed. A has the values above or in addn. is CH(OCH2C6H5); R1, R2, R3 = amino-protective gps. of alkoxycarbonyl, benzyloxycarbonyl or benzyl type.</p> |
申请人 |
FOURNIER INDUSTRIE ET SANTE, PARIS, FR |
发明人 |
RENAUT, PATRICE, F-21121 HAUTEVILLE-LES-DIJON, FR;LEBRETON, LUC, F-21000 DIJON, FR;DUTARTRE, PATRICK, F-21110 LONGCHAMP, FR;DERREPAS, PHILIPPE, F-21410 AGEY, FR;SAMRETH, SOTH, F-21600 LONGVIC, FR |