发明名称 |
Antimigraine-4-pyrimidinyl and pyridinyl derivatives of indol-3yl-alkyl piperazines. |
摘要 |
A series of novel alkoxypyridin-4-yl and alkoxypyrimidin-4-yl derivatives of indol-3-ylalkylpiperazines of formula I are intended to be useful agents for alleviation of vascular headache on the basis of their potent affinity and agonist activity at 5-HT1D binding sites. <CHEM> n |
申请公布号 |
PH30988(A) |
申请公布日期 |
1997.12.23 |
申请号 |
PH19270000454 |
申请日期 |
1992.12.15 |
申请人 |
BRISTOL-MYERS SQUIBB CO. |
发明人 |
SMITH, DAVID, W.;YEVICH, JOSEPH, P.;WILLIAMS ANDREW;RUEDIGER, EDWARD, H.;COMBRINK KEITH DEAN;PEARCE BRADLEY CLYDE |
分类号 |
A61K31/495;A61K31/40;A61K31/44;A61K31/505;A61K31/506;A61P25/04;A61P25/06;C07D209/10;C07D213/65;C07D239/36;C07D241/04;C07D401/12;C07D401/14;C07D403/12;C07D403/14 |
主分类号 |
A61K31/495 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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