发明名称 Tachykinin antagonists
摘要 The invention concerns tachykinin antagonists. The compounds are nonpeptides which have utility in treating disorders mediated by tachykinins. Such disorders are respiratory, inflammatory, gastrointestinal, ophthalmic, allergies, pain, vascular, diseases of the central nervous system, and migraine. Methods of preparing compounds and novel intermediates are also included. The compounds are expected to be especially useful in asthma and rheumatoid arthritis.
申请公布号 US5594022(A) 申请公布日期 1997.01.14
申请号 US19940344064 申请日期 1994.11.29
申请人 WARNER-LAMBERT COMPANY 发明人 HORWELL, DAVID C.;HOWSON, WILLIAM;PRITCHARD, MARTYN C.;ROBERTS, EDWARD;REES, DAVID C.
分类号 C07D333/68;A61K31/27;A61K31/38;A61K31/381;A61K31/40;A61K31/403;A61K31/404;A61K31/44;A61K31/4427;A61K31/443;A61K31/4433;A61K49/00;A61P1/00;A61P9/10;A61P11/00;A61P11/06;A61P25/00;A61P25/04;A61P27/02;A61P27/14;A61P29/00;A61P35/00;A61P37/08;A61P43/00;C07C271/18;C07C271/22;C07D209/20;C07D209/30;C07D231/56;C07D333/60;C07D401/12;C07D405/12;C07D405/14;C07D409/12;C07D417/12;(IPC1-7):C07D209/12;C07D403/12;C07D407/12 主分类号 C07D333/68
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