发明名称 |
N,N'-CARBONYL-BIS-(4-ETHYL-2,3-DIOXO)-PIPERAZINE, PROCESS FOR THE PREPARATION THEREOF AND USE THEREOF |
摘要 |
A new compound called N,N'-carbonyl-bis-(4-ethyl-2,3-dioxo)-piperazine of Formula I <IMG> (I) A process for the preparation thereof based on the reaction of 4-ethyl-2,3-dioxo-piperazine or a trimethylsilyl derivative thereof with carbonyl chloride or a derivative thereof. The use of the compound of Formula I as an intermediate in the preparation of compounds of Formula II <IMG> (II) where R is a radical, substituted in alpha position, of a molecule of an acid selected from the group formed by phenylacetic acid, p-hydroxy phenylacetic acid, a 6 (phenylacetamido)-penicillanic acid and a 7-(phenyl-acetamido)-cephalosporanic acid.
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申请公布号 |
CA1338624(C) |
申请公布日期 |
1996.10.01 |
申请号 |
CA19880582522 |
申请日期 |
1988.11.08 |
申请人 |
BIOCHEMIE, S.A. |
发明人 |
CASTELLVI, JUAN CABRE;MESEGUER, JOSE DIAGO;BIANCHINI, ASUNCION ESTEVE;PADRO, CARLOS E. LENHARDT;PITARCH, ESTEVE SANS |
分类号 |
C07D241/08;C07D499/00;C07D499/68;C07D501/20;C07D501/36;(IPC1-7):C07D241/08;C07D499/70 |
主分类号 |
C07D241/08 |
代理机构 |
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