| 发明名称 |
PROCESS TO MAKE HIV PROTEASE INHIBITOR FROM 2(S)-4-PICOLYL-2-PIPERAZINE-t-BUTYLCARBOXAMIDE |
| 摘要 |
<p>A process for making a clinically efficacious HIV protease inhibitor eliminates one step in its synthesis, by an alternative convergent synthesis using 2(S)-4-picolyl-2-piperazine-t-butylcarboxamide as an intermediate; as indicated above.</p> |
| 申请公布号 |
WO9628439(A1) |
申请公布日期 |
1996.09.19 |
| 申请号 |
WO1996US02556 |
申请日期 |
1996.03.11 |
| 申请人 |
MERCK & CO., INC. |
发明人 |
ASKIN, DAVID;ENG, KAN, K.;REIDER, PAUL;VOLANTE, RALPH, P. |
| 分类号 |
C07D401/06;(IPC1-7):C07D401/06;A61K31/495 |
主分类号 |
C07D401/06 |
| 代理机构 |
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代理人 |
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| 主权项 |
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