发明名称 |
BICYCLING LACTAM INHIBITOR OF INTERLEUKIN-1-BETA CONVERTING ENZYME |
摘要 |
Disclosed are compounds, compositions, and methods for inhibiting interleukin1.beta. protease activity, having formula (A), wherein Y = (a) or (b) or (c), Z = various bicyclic lactams with a bridgehead nitrogen.
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申请公布号 |
CA2192360(A1) |
申请公布日期 |
1995.12.14 |
申请号 |
CA19952192360 |
申请日期 |
1995.06.08 |
申请人 |
SANOFI WINTHROP, INC. |
发明人 |
SCHMIDT, STANLEY J.;MORGAN-ROSS, TINA;DOLLE, ROLAND E.;CHATURVEDULA, PRASAD V. |
分类号 |
C07D487/04;A61K31/535;A61K31/55;A61K38/00;A61P29/00;A61P35/00;A61P37/06;A61P43/00;C07D471/04;C07D513/04;C07K5/02;C07K5/06;C07K5/078;(IPC1-7):C07D487/04;A61K31/435;A61K31/495;C07F9/656;A61K31/675 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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