发明名称 4-acylthio azetidinones
摘要 There is provided a process for preparing a compound of formula (I) <CHEM> wherein R is H or a hydroxy protecting group, R2 is an organic residue and R3 is H or a nitrogen protecting group, which process comprises reacting together a compound of formula (II) <CHEM> wherein R1 is a C1-C4 alkyl or a phenyl group, R and R3 are as defined above, a compound of formula (III) <CHEM> wherein R2 is as defined above and X is a cation or a silicon-containing residue, and a salt of a group IIa, IIb or transition element. The compounds of formula (I) are intermediates in the synthesis of penem antibiotics.
申请公布号 AU4325593(A) 申请公布日期 1994.01.04
申请号 AU19930043255 申请日期 1993.06.14
申请人 FARMITALIA CARLO ERBA S.R.L. 发明人 WALTER CABRI;ILARIA CANDIANI;FRANCO ZARINI;ANGELO BEDESCHI
分类号 C07D205/09;C07D401/12;C07D405/12;C07D499/88;C07D499/897;C07F7/18 主分类号 C07D205/09
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