| 发明名称 |
SUBSTITUTED AMINE DERIVATIVES OF PIPERIZINYLCAMPHORSULFONYL OXYTOCIN ANTAGONISTS |
| 摘要 |
TITLE OF THE INVENTION SUBSTITUTED AMINE DERIVATIVES OF PIPERIZINYLCAMPHORSULFONYL OXYTOCIN ANTAGONISTS Compounds of the formula: and the pharmaceutically acceptable salts thereof, are oxytocin antagonists useful in the treatment of preterm labor, dysmenorrhea and for the stoppage of labor preparatory to cesarean delivery. Also disclosed are pharmaceutical compositions containing these compounds, methods of their use and methods of their preparation.
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| 申请公布号 |
CA2078025(A1) |
申请公布日期 |
1993.03.17 |
| 申请号 |
CA19922078025 |
申请日期 |
1992.09.11 |
| 申请人 |
MERCK & CO., INC. |
发明人 |
ERB, JILL M.;VEBER, DANIEL F.;WILLIAMS, PETER D. |
| 分类号 |
A61K31/495;A61P13/02;A61P15/00;C07D207/16;C07D207/26;C07D207/273;C07D207/277;C07D207/38;C07D207/404;C07D209/08;C07D211/58;C07D211/60;C07D211/62;C07D213/36;C07D213/38;C07D213/64;C07D213/74;C07D213/82;C07D233/54;C07D233/64;C07D233/76;C07D239/02;C07D239/06;C07D239/10;C07D241/08;C07D249/14;C07D257/04;C07D295/16;C07D295/18;C07D295/22;C07D295/26;C07D303/04;C07D303/34;C07D307/33;C07D307/42;C07D309/14;C07D333/24;C07D335/02;C07D403/12;C07D453/02;(IPC1-7):C07D295/26;C07D401/12;C07D405/12;C07D409/12 |
主分类号 |
A61K31/495 |
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