发明名称 |
Antipsychotic 3-piperazinyl-benzazole derivatives. |
摘要 |
Novel 3-piperazinyl-1,2-benzazoles of formula <CHEM> wherein Q is a radical of formula <CHEM> R is hydrogen or C1-6alkyl; R<1> and R<2> are hydrogen, halo, hydroxy, C1-6alkyloxy or C1-6alkyl; X is O, S or NR<3>; the pharmaceutically acceptable acid addition salts and possible stereochemically isomeric forms thereof, which compounds are antipsychotic agents; pharmaceutical compositions containing such compounds as an active ingredient and methods of preparing said compounds and pharmaceutical compositions.
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申请公布号 |
EP0353821(A2) |
申请公布日期 |
1990.02.07 |
申请号 |
EP19890201981 |
申请日期 |
1989.07.28 |
申请人 |
JANSSEN PHARMACEUTICA N.V. |
发明人 |
KENNIS, LUDO EDMOND JOSEPHINE;VANDENBERK, JAN;MERTENS, JOSEPHUS CAROLUS |
分类号 |
C07D417/04;A61K31/496;A61K31/505;A61K31/517;A61K31/54;A61P25/00;A61P25/02;A61P43/00;C07D231/56;C07D261/20;C07D275/04;C07D403/12;C07D413/12;C07D417/12;C07D471/04;C07D498/04;C07D513/04 |
主分类号 |
C07D417/04 |
代理机构 |
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地址 |
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