发明名称 |
6-FLUORO-1,4-DIHYDRO-4-OXO-7-(4-PYRIDYL)-1,8- NAPHTHYRIDINE-3 CARBOXYLIC ACID COMPOUNDS |
摘要 |
<p>The invention provides for novel 7-(4-pyridyl)-1,8-naphthyridine derivatives of the formula (I) (I) wherein R1 is a hydrogen atom, an ethyl or vinyl group, and R2 is a hydrogen atom or a lower alkyl group having 1 to 6 carbon atoms, and processes for their preparation. The compounds of the invention exhibit superior antibacterial activity against Gram-positive bacteria such as Staphylococcus aureus, Gram-negative bacteria such as Escherichia coli and glucose-non-fermenters including Pseudomonas aeuroginosa.</p> |
申请公布号 |
CA1250846(A) |
申请公布日期 |
1989.03.07 |
申请号 |
CA19830433526 |
申请日期 |
1983.07.29 |
申请人 |
DAINIPPON PHARMACEUTICAL CO., LTD.;LABORATOIRE ROGER BELLON |
发明人 |
MATSUMOTO, JUN-ICHI;NISHIMURA, YOSHIRO;NAKAMURA, SHINICHI |
分类号 |
A61K31/44;A61P31/04;C07D471/04;(IPC1-7):C07D471/04 |
主分类号 |
A61K31/44 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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