摘要 |
<p>There are described novel pyrrolo[1,2-b][1,2,5]triazepines of the general formula <IMAGE> (I) where R is hydrogen, loweralkyl, loweralkylaminoloweralkyl or diloweralkylaminoloweralkyl; X is hydrogen, halogen (fluorine, chlorine, bromine or iodine), trifluoromethyl or nitro; and Y is hydrogen, halogen or loweralkyl. Also described are derivatives of 1-amino-2-benzoylpyrrole having the general formula <IMAGE> (II) where R, X and Y are as defined above, and R1 is hydrogen, <IMAGE> <IMAGE> <IMAGE> <IMAGE> +TR <IMAGE> Compounds I and II are useful as analgesic, anxiolytic and/or anticonvulsant agents, and many of Compounds II are useful as intermediates for synthesizing Compounds I.</p> |