发明名称 FRAMSTAELLNING AV 3-ACYLAMINOIMIDAZOL/1,2-C/PYRIDINDERIVAT OCH DERAS TERAPEUTISKA TILLAEMPNING.
摘要 Compounds which are imidazo[1,2-a]pyridine derivatives of general formula (I) <IMAGE> (I) in which each of X1, X2, X3, independently of each other, is hydrogen, halogen, C1-C4 alkyl, methoxy, methylthio, ethylthio, methylsulphonyl, nitro, amino, methylamino, dimethylamino, acetylamino or diacethylamino, Y is hydrogen, chlorine or methyl, R1 is hydrogen, C1-C4 alkyl or benzyl, R2 is C1-C6 alkyl, cyclohexyl, trichloromethyl, 1-propenyl, allyl, phenyl, 4-chlorophenyl or benzyl, or R1 and R2 together represent a divalent C3-C5 alipathic group and their pharmaceutically acceptable acid salts have anxiolytic, sleep-inducing, hypnotic, anticonvulsant, analgesic and anti-ulcer properties.
申请公布号 FI853026(L) 申请公布日期 1986.02.08
申请号 FI19850003026 申请日期 1985.08.06
申请人 SYNTHELABO 发明人 GEORGE, PASCAL;GIRON, CLAUDIE
分类号 C07D487/04;A61K31/435;A61K31/44;A61P25/08;A61P25/20;A61P25/28;C07D471/04 主分类号 C07D487/04
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