发明名称 Pyridinyl-substituted benzimidazoles and quinoxalines.
摘要 <p>Pyridinyl-benzimidazoles and quinoxalines which may be useful as thromboxane A2 (TXA2) synthetase inhibitors, and which have formula I or II &lt;CHEM&gt; wherein Z1 is 4-pyridinyl, 3-pyridinyl or (C1-4 alkyl)-3-pyridinyl, X1 is C1-3 n-alkylene, -O-, -CH2O- or -OCH2-, m is from zero to 4 and R7 is -CH2OH, -CHO or optionally esterified or salified carboxyl. </p>
申请公布号 EP0104727(A1) 申请公布日期 1984.04.04
申请号 EP19830304436 申请日期 1983.08.01
申请人 THE UPJOHN COMPANY 发明人 NELSON, NORMAN ALLAN
分类号 C12N9/99;A61K31/44;A61K31/4409;A61K31/4418;A61K31/4427;A61K31/495;A61P1/04;A61P7/02;A61P9/12;A61P29/00;A61P35/00;A61P43/00;C07D213/40;C07D213/53;C07D401/06;C07D401/12;(IPC1-7):07D401/06;61K31/415;61K31/495;61K31/44;07D401/12 主分类号 C12N9/99
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