发明名称 6-PHENYL-8-BROMO-4H-S-TRIAZOLO-(3,4C)-THIENO-(2,3E)-1,4-DIAZEPINES AND SALTS THEREOF
摘要 Compounds of the formula <IMAGE> wherein R1 is hydrogen, chlorine, bromine or alkyl of 1 to 4 carbon atoms; R2 is hydrogen, fluorine, chlorine, bromine, nitro or trifluoromethyl; and R3 is chlorine, bromine, alkoxy of 1 to 3 carbon atoms, alkylmercapto of 1 to 3 carbon atoms, cycloalkyl of 3 to 6 carbon atoms, cycloalkenyl of 3 to 6 carbon atoms, or a saturated or unsaturated 5- to 6-membered heterocycle comprising an oxygen, sulfur or nitrogen heteroatom, where a substitutable nitrogen heteroatom may optionally have a lower akyl substituent attached thereto; and non-toxic, pharmacologically acceptable acid addition salts thereof; the compounds as well as their salts are useful as tranquilizers, muscle-relaxants and anticonvulsants.
申请公布号 US4094984(A) 申请公布日期 1978.06.13
申请号 US19770839792 申请日期 1977.10.06
申请人 BOEHRINGER INGELHEIM GMBH 发明人 WEBER, KARL-HEINZ;BAUER, ADOLF;DANNEBERG, PETER;KUHN, FRANZ JOSEF
分类号 A61K31/55;A61K31/551;A61P25/00;C07D333/36;C07D495/04;C07D495/14;(IPC1-7):A61K31/55 主分类号 A61K31/55
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