发明名称 Optically active azole compounds and their production
摘要 An optically active azole compound of the formula (I): <IMAGE> (I) wherein R1 and R2 are independently a hydrogen atom, a halogen atom, a haloalkyl group, a haloalkoxy group or an optionally substituted nitrogen-containing heterocyclic group; R3 is a hydrogen atom or an acyl group; Q is CH or N; <IMAGE> is a nitrogen-containing aromatic five-membered heterocyclic group having at least two adjacent nitrogen atoms as the ring-constituting atoms which may be substituted, or an aromatic condensed heterocyclic group having two or more nitrogen atoms as the ring-constituting atoms which may be substituted; and (R) shows that the carbon atom marked with (R) has R-configuration; provided that either of R1 and R2 is an optionally substituted nitrogen-containing heterocyclic group when <IMAGE> is an 1H-1,2,4-triazol-1-yl group, or a salt thereof, which is useful as an antifungal agent.
申请公布号 US5495024(A) 申请公布日期 1996.02.27
申请号 US19940302411 申请日期 1994.09.08
申请人 TAKEDA CHEMICAL INDUSTRIES LTD. 发明人 ITOH, KATSUMI;OKONOGI, KENJI;TAMURA, NORIKAZU
分类号 C07D249/08;C07D521/00;(IPC1-7):C07D249/08;C07D405/06 主分类号 C07D249/08
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