发明名称 |
BIS-SULFONAMID-HYDROXYETHYLAMINO-DERIVATE ALS INHIBITOREN RETROVIRALER PROTEASEN |
摘要 |
Bis-sulfonamido hydroxyethylamino compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to retroviral protease inhibiting compounds of the formula: <CHEM> or a pharmaceutically acceptable salt, prodrug or ester thereof, wherein the variables are as defined herein. |
申请公布号 |
DE69637380(D1) |
申请公布日期 |
2008.02.07 |
申请号 |
DE1996637380 |
申请日期 |
1996.01.18 |
申请人 |
G.D. SEARLE LLC |
发明人 |
FRESKOS, JOHN N.;GETMAN, DANIEL P.;TALLEY, JOHN J.;SIKORSKI, JAMES A. |
分类号 |
C07D295/08;C07D295/22;A61K31/18;A61K31/185;A61K31/195;A61K31/335;A61K31/336;A61K31/34;A61K31/341;A61K31/343;A61K31/357;A61K31/36;A61K31/38;A61K31/381;A61K31/40;A61K31/4025;A61K31/415;A61K31/4184;A61K31/42;A61K31/423;A61K31/425;A61K31/428;A61K31/443;A61K31/445;A61K31/454;A61K31/495;A61K31/496;A61K31/535;A61K31/5355;A61K31/5375;A61K31/5377;A61P31/12;A61P43/00;C07C311/29;C07C311/38;C07D213/38;C07D233/54;C07D233/61;C07D235/06;C07D235/26;C07D235/30;C07D235/32;C07D263/54;C07D277/66;C07D277/82;C07D295/12;C07D295/26;C07D303/36;C07D307/14;C07D307/79;C07D317/62;C07D319/18;C07D333/34;C07D405/12;C07D417/12 |
主分类号 |
C07D295/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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