发明名称 N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES
摘要 The novel compounds of formula (I), wherein R1, R2, R2', R2'', R3, R4, R5, R5', R5'', R5''', R'''', X, Y, U, V and W have the meanings given in patent claim no. 1, are inhibitors of the coagulation factors Xa and VIIa and can be used for treating thromboses, myocardial infarction, arteriosclerosis, inflammations, apoplexy, angina pectoris, restenosis following angioplasty, intermittent claudication, tumours, tumour diseases and/or tumour metastases.
申请公布号 PL358585(A1) 申请公布日期 2004.08.09
申请号 PL20010358585 申请日期 2001.07.03
申请人 MERCK PATENT GMBH 发明人 JURASZYK HORST;DORSCH DIETER;MEDERSKI WERNER;TSAKLAKIDIS CHRISTOS;BARNES CHRISTOPHER;GLEITZ JOHANNES
分类号 A61K31/18;A61K31/277;A61K31/4245;A61P7/02;A61P9/00;A61P9/10;A61P29/00;A61P35/00;A61P35/04;C07B61/00;C07C311/46;C07D211/66;C07D213/40;C07D271/06;C07D309/14;C07D335/02;C07D401/12;C07D405/12;C07D409/12;C07D413/12 主分类号 A61K31/18
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