发明名称 Ketoheteroarylpiperdine and -piperazine derivatives as fungicides
摘要 Ketoheteroarylpiperidine and -piperazine derivatives of the formula (I),; in which the symbols A, L1, G, X, Y, T and R1 have the meanings given in the description and agrochemically active salts thereof and their use for controlling phytopathogenic harmful fungi and also processes for preparing compounds of the formula (I).
申请公布号 US9357779(B2) 申请公布日期 2016.06.07
申请号 US201313800521 申请日期 2013.03.13
申请人 Bayer Intellectual Property GmbH 发明人 Cristau Pierre;Hoffmann Sebastian;Kluth Joachim;Seitz Thomas;Tsuchiya Tomoki;Wasnaire Pierre;Benting Jürgen;Wachendorff-Neumann Ulrike
分类号 A01N43/40;C07D419/04;A01P3/00;A01N43/78;C07D417/12;C07D417/14 主分类号 A01N43/40
代理机构 Sterne, Kessler, Goldstein & Fox P.L.L.C. 代理人 Sterne, Kessler, Goldstein & Fox P.L.L.C.
主权项 1. A method for controlling phytopathogenic harmful fungi, the method comprises administering an effective amount of at least one compound of formula (I′), wherein: A represents phenyl which may contain up to two substituents, wherein the substituents independently of one another are selected from R2, and R2 represents: methyl, ethyl, iodine, chlorine, bromine, fluorine, methoxy, ethoxy, difluoromethyl, or trifluoromethyl, or A represents pyrazol-1-yl which, may contain up to two substituents at carbon, wherein the substituents independently of one another are selected from R3, and R3 represents methyl, difluoromethyl, or trifluoromethyl, T is selected from the group consisting of *—C(═O)CH2—#, *—C(═O)CH2C(CH3)2—#, *—C(═O)CH2CH2—#, *—C(═O)CH═CH—#, *—C≡CC(═O)—#, *—CH═CHC(═O)—#, *CH2CH2C(═O)—#, *—C(═NOCH3)CH2—#, *—CH═CHC(NOH)—#, *—C(Cl)═CHC(═O)—#, and *—CH(CH3)CH2C(═O)—#, where the bond identified by * is attached directly to G and where the bond identified by # is attached directly to R1, R1 is selected from the group consisting of R1a, R1b, R1 c, R1d, R1e, and R1f, wherein R1a represents 1,1-dimethylethyl, R1b represents cyclohexyl, cyclopentyl, 2-methylcyclohexyl, 3-methylcyclohexyl, or 4-methylcyclohexyl, R1c represents cyclohex-3-en-1-yl or cyclohex-2-en-1-yl, R1d represents phenyl that may contain up to two substituents, wherein the substituents independently of one another are selected from R12, and R12 represents:chlorine, fluorine, bromine, iodine, methyl, methoxy, ethoxy, trifluoromethyl, difluoromethyl, 2-propenyloxy, 2-propynyloxy or phenyl, R1e represents naphthalen-1-yl, naphthalen-2-yl, 1,2,3,4-tetrahydronaphthalen-1-yl, 1,2,3,4-tetrahydronaphthalen-2-yl, 5,6,7,8-tetrahydronaphthalen-1-yl, 5,6,7,8-tetrahydronaphthalen-2-yl, decalin-1-yl, decalin-2-yl, 1H-inden-1-yl, 1H-inden-2-yl, 1H-inden-3-yl, 1H-inden-4-yl, 1H-inden-5-yl, 1H-inden-6-yl, 1H-inden-7-yl, indan-1-yl, indan-2-yl, indan-3-yl, indan-4-yl, or indan-5-yl, R1f represents furan-2-yl, furan-3-yl, thiophen-2-yl, thiophen-3-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, pyrrol-1-yl, pyrrol-2-yl, pyrrol-3-yl, oxazol-2-yl, oxazol-4-yl, oxazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl, pyrazol-1-yl, pyrazol-3-yl, pyrazol-4-yl, imidazol-1-yl, imidazol-2-yl, imidazol-4-yl, 1,2,3-triazol-1-yl, 1,2,3-triazol-2-yl, 1,2,3-triazol-4-yl, 1,2,4-triazol-1-yl, 1,2,4-triazol-3-yl, 1,2,4-triazol-4-yl, pyridin-2-yl, pyridin-3-yl, pyridin-4-yl pyridazin-3-yl, pyridazin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl, or pyrimidin-5-yl, or an agrochemically active salt thereof.
地址 Monheim DE