| 摘要 |
These are new azol derivs. of formula (I), which are useful for eumycetes therapeutics. In the formula, Q is C or N; Ar is 2,4-difluorophenyl, 2,4-dichlorophenyl, 4-fluorophenyl, 4-chlorophenyl, 4-trifluorophenyl, 2-fluoro-4-chlorophenyl, 4-bromophenyl; R1 and R2 is H, methyl, ethyl, propyl, isopropyl or cyclopropyl, respectively; R3 is H, Cl, Br, I, methyl, ethyl, propyl, butyl, hexyl, phenyl, naphthyl, 3,4-dimethoxyphenyl, diethylamino, 3,4,5-trimethoxyphenyl, 2-chlorophenyl, 2-bromophenyl, 2-fluorophenyl, 2-nitrophenyl, 4-hydroxyphenyl, 4-aminophenyl, 2,4-dichlorophenyl, 2-chloro-6-fluorophenyl, 2,4-difluorophenyl, 3-fluorophenyl, 3-bromophenyl, 3-chlorophenyl, 4-bromophenyl, 4-fluorophenyl, 4-chlorophenyl, 2,6-dichlorophenyl, 3,4-dichlorophenyl, 2,5-dichlorophenyl, 2,6-difluorophenyl, 3,4-difluorophenyl, 3,4-(methylenedioxy)phenyl, 2-pyridyl, 3-pyridyl or 4-pyridyl; R4 is H, Cl, F, or I; N is an integer of 0-2.
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