| 摘要 |
The present invention discloses benzo-heterocyclic compounds substituted by aminoalkyl groups, of formula (See Formula) wherein R is a group of formula (See Formula) T is H, alkyl, halogen, N(R2,R21), CONH2, CN, NO2, CF3, OH or alkyl-(O or S); R2 and R21 are alkyl or H and Q is cycloalkyl, optionally substituted phenyl or alkyl-alkenyl or optionally substituted by OH, or wherein one of the two substituents R and T is halogen or H and the other one is H, alkyl, halogen, N(R2,R21), CONH2, CN, NO2, CF3, OH or alkyl-(O or S) and Q is a group of formula (See Formula) A1 is alkyl or alkenyl and A2 is cycloalkyl, cycloalkyl-alkyl or an alkyl group or optionally substituted alkenyl or A1 and A2 together are an alkylen or alkenilene, L1 is a L group, directly linked to the benzo group or by NH or N-(alkyl or alkanoyl), L2 is an alkylen or alkenilene group or else a (cycloalkylen)-alkylen group, M dotted linkage is optional, M is a group of 2 or 3 links containing a O or S atom or a group S(O), S(O)2 or C(O) and/or until two N atoms or groups N(R6) and/or until two groups C(R6) O CH(R6), but which contains in total at least an optionally substituted heteroatom and R6 is H or alkyl, and acid addition salts therefrom.
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