发明名称 |
Inhibitors of histone deacetylase |
摘要 |
This invention relates to five specific N-hydroxybenzamide compounds for the inhibition of histone deacetylase: N-hydroxy-4-(5-(p-tolyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl)benzamide; N-hydroxy-4-(5-(3-methoxyphenyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl)benzamide; N-hydroxy-4-(5-(4-(trifluoromethyl)pyridin-2-yl)-2,5-diazabicyclo[2.2.1]heptan-2-yl)benzamide; 4-(benzo[b]thieno[2,3-f][1,4]oxazepin-10-yl)-N-hydroxybenzamide; and 4-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-hydroxybenzamide. |
申请公布号 |
EP2966078(A3) |
申请公布日期 |
2016.03.09 |
申请号 |
EP20140194168 |
申请日期 |
2007.10.26 |
申请人 |
METHYLGENE INC.;FORUM PHARMACEUTICALS INC. |
发明人 |
DEZIEL, ROBERT;LEIT, SILVANA;BEAULIEU, PATRICK;CHANTIGNY, YVES, ANDRE;MANCUSO, JOHN;TESSIER, PIERRE;SHAPIRO, GIDEON;CHESWORTH, RICHARD;SMIL, DAVID |
分类号 |
C07D498/04;A61K31/4995;A61K31/55;A61K31/553;A61P25/00;C07D223/28;C07D487/08 |
主分类号 |
C07D498/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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