发明名称 1 -(CYCLOPENT-2-EN-1 -YL)-3-(2-HYDROXY-3-(ARYLSULFONYL)PHENYL)UREA DERIVATIVES AS CXCR2 INHIBITORS
摘要 <p>The invention relates to 1-(3-sulfonylphenyl)-3-(cyclopent-2-en-1-yl)urea derivatives, and their use in treating or preventing diseases and conditions mediated by the CXCR2 receptor. In addition, the invention relates to compositions containing the derivatives and processes for their preparation.</p>
申请公布号 WO2015181186(A1) 申请公布日期 2015.12.03
申请号 WO2015EP61618 申请日期 2015.05.27
申请人 GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENTLIMITED 发明人 CHEN, WEICHUN;IGBOKO, EBERE F;LIN, XICHEN;LU, HONGFU;REN, FENG;WREN, PAUL BRYAN;XU, ZHONGMIAO;YANG, TING;ZHU, LINGDONG
分类号 C07C211/56;A61K31/17;A61P11/00;A61P29/00;C07C275/30;C07D207/10;C07D211/54;C07D213/34;C07D233/64;C07D239/26;C07D295/135;C07D305/06;C07D307/18;C07D309/08;C07D471/04;C07D487/04 主分类号 C07C211/56
代理机构 代理人
主权项
地址