主权项 |
化合物,其为:{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基}‑(4‑氟‑苯基)‑甲酮;{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基}‑异噻唑‑3‑基‑甲酮;{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基}‑(5‑哌啶‑1‑基‑吡嗪‑2‑基)‑甲酮;{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基}‑(6‑苯氧基‑吡啶‑3‑基)‑甲酮;5‑乙基‑2‑氟‑4‑{3‑[5‑(6‑吗啉‑4‑基‑吡啶‑3‑磺酰基)‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基]‑1H‑吲唑‑6‑基}‑苯酚;5‑乙基‑2‑氟‑4‑{3‑(5‑(6‑苯氧基‑吡啶‑3‑磺酰基)‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基]‑1H‑吲唑‑6‑基}‑苯酚;(5‑氯‑吡啶‑2‑基)‑{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑4,5,7,8‑四氢‑1H‑咪唑并[4,5‑d]氮杂<img file="FDA0000719572850000011.GIF" wi="62" he="71" />‑6‑基}‑甲酮;2‑{2‑[6‑{2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑4,5,7,8‑四氢‑1H‑咪唑并[4,5‑d]氮杂<img file="FDA0000719572850000012.GIF" wi="62" he="71" />‑6‑羰基}‑异烟腈;{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑4,5,7,8‑四氢‑1H‑咪唑并[4,5‑d]氮杂<img file="FDA0000719572850000013.GIF" wi="62" he="76" />‑6‑基}‑(4‑氟‑苯基)‑甲酮;{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑4,5,7,8‑四氢‑1H‑咪唑并[4,5‑d]氮杂<img file="FDA0000719572850000014.GIF" wi="62" he="71" />‑6‑基}‑异噻唑‑3‑基‑甲酮;5‑乙基‑2‑氟‑4‑{3‑[5‑(4‑氟‑苯磺酰基)‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基]‑1H‑吲唑‑6‑基}‑苯酚;{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基}‑[5‑(2‑氟‑苯氧基)‑吡嗪‑2‑基]‑甲酮;4‑[3‑(6‑苯甲基‑1,4,5,6,7,8‑六氢‑咪唑并[4,5‑d]氮杂<img file="FDA0000719572850000015.GIF" wi="62" he="76" />‑2‑基)‑1H‑吲唑‑6‑基]‑5‑乙基‑2‑氟‑苯酚;(5‑氯‑吡啶‑2‑基)‑{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基}‑甲酮;5‑{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑羰基}‑吡啶‑2‑甲腈;5‑{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑4,5,7,8‑四氢‑1H‑咪唑并[4,5‑d]氮杂<img file="FDA0000719572850000021.GIF" wi="62" he="80" />‑6‑羰基}‑吡啶‑2‑甲腈;5‑乙基‑2‑氟‑4‑[3‑(5‑喹啉‑6‑基甲基‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基)‑1H‑吲唑‑6‑基]‑苯酚;5‑乙基‑2‑氟‑4‑{3‑[5‑(4‑羟基‑苯甲基)‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基]‑1H‑吲唑‑6‑基}‑苯酚;5‑乙基‑2‑氟‑4‑{3‑[5‑(3‑羟基‑苯甲基)‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基]‑1H‑吲唑‑6‑基}‑苯酚;4‑{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基甲基}‑吡啶‑2‑甲腈;5‑乙基‑2‑氟‑4‑{3‑[5‑(3‑甲氧基‑苯甲基)‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基]‑1H‑吲唑‑6‑基}‑苯酚;5‑乙基‑2‑氟‑4‑[3‑(5‑喹啉‑3‑基甲基‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基)‑1H‑吲唑‑6‑基]‑苯酚;5‑乙基‑2‑氟‑4‑{3‑[5‑(6‑苯氧基‑吡啶‑3‑基甲基)‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基]‑1H‑吲唑‑6‑基}‑苯酚;5‑乙基‑2‑氟‑4‑{3‑[5‑(3,4,5,6‑四氢‑2H‑[1,2’]联吡啶‑5'‑基甲基)‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基]‑1H‑吲唑‑6‑基}‑苯酚;3‑{2‑[6‑(2‑乙基‑5‑氟‑4‑羟基‑苯基)‑1H‑吲唑‑3‑基]‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基甲基}‑吡啶‑2‑甲腈;5‑乙基‑2‑氟‑4‑{3‑[5‑(4‑氟‑苯甲基)‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基]‑1H‑吲唑‑6‑基)‑苯酚;5‑乙基‑2‑氟‑4‑[3‑(5‑[1,8]二氮杂萘‑2‑基甲基‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基)‑1H‑吲唑‑6‑基]‑苯酚;(2‑{6‑[5‑氟‑4‑羟基‑2‑(2,2,2‑三氟‑乙基)‑苯基]‑1H‑吲唑‑3‑基}‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基)‑(5‑哌啶‑1‑基‑吡嗪‑2‑基)‑甲酮;(2‑{6‑[5‑氟‑4‑羟基‑2‑(2,2,2‑三氟‑乙基)‑苯基]‑1H‑吲唑‑3‑基}‑1,4,6,7‑四氢‑咪唑并[4,5‑c]吡啶‑5‑基)‑(4‑氟‑苯基)‑甲酮;或4‑[3‑(5‑苯甲基‑4,5,6,7‑四氢‑1H‑咪唑并[4,5‑c]吡啶‑2‑基)‑1H‑吲唑‑6‑基]‑2‑氟‑5‑(2,2,2‑三氟‑乙基)‑苯酚;或其药学上可接受的盐。 |