发明名称 |
SUBSTITUTED 4-{3-[6-AMINO-9-(3,4-DIHYDROXY-TETRAHYDRO-FURAN-2-YL) -9H-PURIN-2-YL]-PROP-2-YNYL}-PIPERIDINE-1-CARBOXYLIC ACID ESTERS AS A2AR AGONISTS. |
摘要 |
<p>The present invention provides substituted 4-{3-[6-amino-9-(3,4-dihydroxy-tetrahydro-furan-2-yl)-9H-purin- 2-yl]-prop-2-ynyl}-piperidine-1-carboxylic acid esters and pharmaceutical compositions containg the same that are selective agonists of A2A adenosine receptors (ARs). These compounds and compositions are useful as pharmaceutical agents.</p> |
申请公布号 |
MX2010006645(A) |
申请公布日期 |
2010.10.05 |
申请号 |
MX20100006645 |
申请日期 |
2008.12.20 |
申请人 |
PGXHEALTH, LLC |
发明人 |
ROBERT THOMPSON;ANTHONY BEAUGLEHOLE;FRANK SCHMIDTMANN;JAYSON RIEGER |
分类号 |
A01N43/90;A61K31/52;A61K31/7042;A61K31/7076;A61K49/06;A61K49/10;A61P37/08;C07H19/167 |
主分类号 |
A01N43/90 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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