发明名称 PIPERAZINE DERIVATIVES AS HIV PROTEASE INHIBITORS
摘要 Provided are compounds of Formula (I), pharmaceutical compositions comprising the same, and their use in the inhibition of HIV protease, the inhibition of HIV replication, the prophylaxis of infection by HIV, the treatment of infection by HIV, and the prophylaxis, treatment, and delay in the onset or progression of AIDS.
申请公布号 WO2015135091(A1) 申请公布日期 2015.09.17
申请号 WO2014CN00227 申请日期 2014.03.10
申请人 MERCK SHARP & DOHME CORP.;MSD R&D (CHINA) CO., LTD.;WILLIAMS, PETER D.;MCCAULEY, JOHN A.;BUNGARD, CHRISTOPHER J.;BENNETT, DAVID JONATHAN;WADDELL, SHERMAN TIM;MORRIELLO, GREGORI J.;CHANG, LEHUA;DWYER, MICHAEL P.;HOLLOWAY, M. KATHARINE;CRESPO, ALEJANDRO;CHU, XIN-JIE;WISCOUNT, CATHERINE M.;LOUGHRAN, H. MARIE;MANIKOWSKI, JESSE J.;SCHULZ, JURGEN;KEERTIKAR, KARTIK M.;HU, BIN;ZHONG, BIN;JI, TAO 发明人 WILLIAMS, PETER D.;MCCAULEY, JOHN A.;BUNGARD, CHRISTOPHER J.;BENNETT, DAVID JONATHAN;WADDELL, SHERMAN TIM;MORRIELLO, GREGORI J.;CHANG, LEHUA;DWYER, MICHAEL P.;HOLLOWAY, M. KATHARINE;CRESPO, ALEJANDRO;CHU, XIN-JIE;WISCOUNT, CATHERINE M.;LOUGHRAN, H. MARIE;MANIKOWSKI, JESSE J.;SCHULZ, JURGEN;KEERTIKAR, KARTIK M.;HU, BIN;ZHONG, BIN;JI, TAO
分类号 C07D241/00;A61K31/4995;A61P31/18;C07D207/00;C07D213/04 主分类号 C07D241/00
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