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发明名称
制备2,5–双一经取代之胺基一1,3,4一硫杂重氮盐之方法
摘要
申请公布号
TW020222
申请公布日期
1976.03.01
申请号
TW06311378
申请日期
1974.07.02
申请人
氰胺公司
发明人
HARRY LEE LINDSAY;KEITH CHADWICK;MURDOCK;ROBERT BRUCE ANGIER
分类号
A61K31/41;C07D285/135
主分类号
A61K31/41
代理机构
代理人
陈长文 台北巿敦化北路二○一号七楼
主权项
1﹒制备具有下式之化合物的一种方法: 于其中,R为环己基胺基,环戊基胺基或 N─(低级烷基)─1─基者。此方 法之特点为于摄氏40度至130度之温 度,将具有下式之一种化合物 其中之X为溴,与通式(RH)之一种化 合物(其中R之定义如前述)加热2至5 0小时,并于其中回收其生成物,且于需 要时,制备其药物上可接受之酸加成盐类 者。
地址
美国
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