发明名称 A PROCESS FOR THE PREPARATION OF S-[2-[1-(2-ETHYLBUTYL)CYCLOHEXYLCARBONYLAMINO]-PHENYL]-2-METHYLTHIOPIONATE
摘要 <p>The present invention relates to a process for the preparation of S-[2-[1-(2 ethylbutyl)cyclohexylcarbonylamino]-phenyl] 2-methylthiopropionate (see formula I) which is a useful pharmaceutical active compound. The process comprises reacting a compound of formula (II) (see formula II) with isobutyric anhydride and a reducing agent.</p>
申请公布号 CA2764969(C) 申请公布日期 2015.02.03
申请号 CA20102764969 申请日期 2010.06.28
申请人 F. HOFFMANN-LA ROCHE AG 发明人 COSTELLO, DECLAN;HARNETT, GERARD JOHN;HIDBER, PIRMIN;HOFFMANN, URSULA;MCCARTHY, THOMAS;REENTS, REINHARD;SMITH, DENNIS A.;SMYTH, TIMOTHY
分类号 C07C327/30 主分类号 C07C327/30
代理机构 代理人
主权项
地址