发明名称 NOVEL FORMS OF TELAPREVIR
摘要 The invention relates to an amorphous form of telaprevir, its preparation via novel crystalline Form C of telaprevir (also referred to as "crystalline Form C" or "Form C"), and telaprevir compositions comprising said amorphous form and Form C. Furthermore, the present invention relates to the use of said amorphous telaprevir, telaprevir composition and Form C of telaprevir for the preparation of medicaments such as anti-hepatitis C medicaments. Moreover, the present invention relates to pharmaceutical compositions and dosage forms comprising a pharmaceutically effective amount of said novel forms for use in treating patients suffering from hepatitis C virus.
申请公布号 WO2014096343(A1) 申请公布日期 2014.06.26
申请号 WO2013EP77652 申请日期 2013.12.20
申请人 SANDOZ AG 发明人 STEFINOVIC, MARIJAN;LANGES, CHRISTOPH;GRIESSER, ULRICH
分类号 C07D403/12;A61K31/40;A61P31/12;C07K5/087 主分类号 C07D403/12
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