发明名称 SUBSTITUTED PYRIDINE SPLEEN TYROSINE KINASE (Syk) INHIBITORS
摘要 The invention provides certain substituted pyridines of the Formula (I) or pharmaceutically acceptable salts thereof, wherein R1, R2, R3, R4, Rcy,Cy, and t are as defined herein. The invention also provides pharmaceutical compositions comprising such compounds, and methods of using the compounds for treating diseases or conditions mediated by Spleen Tyrosine Kinase (Syk) kinase.
申请公布号 WO2013192098(A1) 申请公布日期 2013.12.27
申请号 WO2013US46151 申请日期 2013.06.17
申请人 MERCK SHARP & DOHME CORP.;MERCK CANADA INC.;HAIDLE, ANDREW, M.;KNOWLES, SANDRA LEE;KATTAR, SOLOMON, D.;DESCHENES, DENIS;BURCH, JASON;ROBICHAUD, JOEL;CHRISTOPHER, MATTHEW;ALTMAN, MICHAEL, D.;JEWELL, JAMES, P.;NORTHRUP, ALAN, B.;BLOUIN, MARC;ELLIS, JOHN, MICHAEL;ZHOU, HUA;FISCHER, CHRISTIAN;SCHELL, ADAM, J.;REUTERSHAN, MICHAEL, H.;TAOKA, BRANDON, M.;DONOFRIO, ANTHONY 发明人 HAIDLE, ANDREW, M.;KNOWLES, SANDRA LEE;KATTAR, SOLOMON, D.;DESCHENES, DENIS;BURCH, JASON;ROBICHAUD, JOEL;CHRISTOPHER, MATTHEW;ALTMAN, MICHAEL, D.;JEWELL, JAMES, P.;NORTHRUP, ALAN, B.;BLOUIN, MARC;ELLIS, JOHN, MICHAEL;ZHOU, HUA;FISCHER, CHRISTIAN;SCHELL, ADAM, J.;REUTERSHAN, MICHAEL, H.;TAOKA, BRANDON, M.;DONOFRIO, ANTHONY
分类号 A61K31/505;A61P35/00 主分类号 A61K31/505
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