发明名称 PROCESS FOR OBTAINING COMPOUNDS DERIVED FROM TETRAHYDRO-BETA-CARBOLINE
摘要 <p>The invention relates to a process for obtaining compounds derived from tetrahydro-beta-carboline, specifically tadalafil and intermediate products from the synthesis, comprising the reaction between piperonal and an alkyl ester of D-tryptophan as a salt, and in the absence of any other component, followed by haloacetylation and a final cyclization with methylamine.</p>
申请公布号 EP2673275(A1) 申请公布日期 2013.12.18
申请号 EP20120704755 申请日期 2012.02.10
申请人 INTERQUIM, S.A. 发明人 BERZOSA RODRIGUEZ, XAVIER;MARQUILLAS OLONDRIZ, FRANCISCO
分类号 C07D471/04;C07D471/14 主分类号 C07D471/04
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