发明名称 |
IMPROVED SYNTHESIS SCHEME FOR LACOSAMIDE |
摘要 |
<p>The present invention is concerned with an improved method of producing (R)-2-acetamido-N-benzyl-3-methoxypropionamide (lacosamide) comprising the 0-methylation of a compound of formula (I) to produce a compound of formula (I I) in a single step reaction.</p> |
申请公布号 |
CA2570598(C) |
申请公布日期 |
2013.12.17 |
申请号 |
CA20052570598 |
申请日期 |
2005.09.30 |
申请人 |
SCHWARZ PHARMA AG |
发明人 |
RIEDNER, JENS;DUNNE, GAVIN |
分类号 |
C07C275/16;C07C231/02;C07C273/18;C07C275/10 |
主分类号 |
C07C275/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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