发明名称 |
METHOD FOR PREPARING 5-CHLORO-N-({(5S)-2-OXO-3-[4-(5,6-DIHYDRO-4H-[1,2,4]TRIAZIN-1-YL)PHENYL]-1,3-OXAZOLIDIN-5-YL}METHYL)THIOPHEN-2-CARBOXAMIDE DERIVATIVE AND INTERMEDIATE USED THEREIN |
摘要 |
Disclosed are: a method for preparing a 5-chloro-N-({(5S)-2-oxo-3-[4-(5,6-dihydro-4H-[1,2,4]triazin-1-yl)phenyl]-1,3-oxazolidin-5-yl}-methyl)thiophene-2-carboxamide derivative, which is a inhibitor of blood coagulation factor Xa, in a high purity and yield; and a novel intermedicate used therein. |
申请公布号 |
EP2451803(A4) |
申请公布日期 |
2013.11.27 |
申请号 |
EP20100797303 |
申请日期 |
2010.07.07 |
申请人 |
GREEN CROSS CORPORATION;LEGOCHEM BIOSCIENCE LTD. |
发明人 |
CHO, YOUNG LAG;CHAE, SANG EUN;KIM, SEONG JIN;SONG, HO YOUNG;PARK, TAE KYO;WOO, SUNG HO;KIM, YONG ZU;LEE, JINHWA;LEE, SUK HO |
分类号 |
C07D403/08;C07D253/06;C07D403/06;C07D409/12;C07D413/14 |
主分类号 |
C07D403/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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