发明名称 |
PREPARATION OF NUCLEOSIDES RIBOFURANOSYL PYRIMIDINES |
摘要 |
<p>The present process provides an improved method for the preparation of 4-amino-1-((2R,3R,4R,5R)-3-fluoro-4-hydroxy-5-hydrox-ymethyl-3-methyl-tetrahydro-furan-2-yl)-1H-pyrimidin-2-one of the formula (IV) which is a potent inhibitor of Hepatitis C Virus (HCV) NS5B polymerase.</p> |
申请公布号 |
SI2084174(T1) |
申请公布日期 |
2013.10.30 |
申请号 |
SI20070031311T |
申请日期 |
2007.10.05 |
申请人 |
GILEAD PHARMASSET LLC;F. HOFFMANN-LA ROCHE AG |
发明人 |
AXT STEVEN D.;SARMA KESHAB;VITALE JUSTIN;ZHU JIANG;ROSS BRUCE;RACHAKONDA SUGUNA;JIN QINGWU;CHUN BYOUNG-KWON |
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