发明名称 |
Hidtil ukendt fremgangsmåde til fremstilling af aminosyrederivater |
摘要 |
<p>The present patent application relates to an alternative process for the preparation of amino derivatives. In particular, the present application relates to an improved process for the manufacture of Lacosamide (LCM), (R)-2-acetamido-N-benzyl-3-methoxypropion-amide, which is useful as an anticonvulsive drug. In a particular aspect, the present invention relates to a process of manufacture of optically enriched (R)-2-acetamido-N-benzyl-3-methoxypropion-amide (I) comprising resolution of 2-acetamido-N-benzyl-3-methoxypropion-amide (II).</p> |
申请公布号 |
DK2352721(T3) |
申请公布日期 |
2013.07.01 |
申请号 |
DK20090799015T |
申请日期 |
2009.11.06 |
申请人 |
UCB PHARMA GMBH |
发明人 |
BOUVY, DIDIER;MERSCHAERT, ALAIN;PINILLA, VERONIQUE;KANZLER, RALF;HAMANN, JOERG;THOMAS, ANTOINE |
分类号 |
C07C231/20;C07C237/06;C07C237/22;C07C237/52 |
主分类号 |
C07C231/20 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|