发明名称 |
Stable Bortezomib Formulations |
摘要 |
Multi-dose formulations for bortezomib are presented in which bortezomib has significantly improved stability. Especially preferred formulations include those in which bortezomib is in a liquid form suitable for injection, wherein the solvent system predominantly comprises propylene glycol. In other preferred aspects, bortezomib is present as a Lewis donor-acceptor complex with a hetero-bifunctional Lewis base.
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申请公布号 |
US2012322763(A1) |
申请公布日期 |
2012.12.20 |
申请号 |
US201213592235 |
申请日期 |
2012.08.22 |
申请人 |
SOPPIMATH KUMARESH;PEJAVER SATISH;PATEL KANAIYALAL R.;DASARADHI LAKKARAJU;SODUM RAMA;DESU HARI;PURI NAVNEET;INNOPHARMA, INC. |
发明人 |
SOPPIMATH KUMARESH;PEJAVER SATISH;PATEL KANAIYALAL R.;DASARADHI LAKKARAJU;SODUM RAMA;DESU HARI;PURI NAVNEET |
分类号 |
A61K31/69 |
主分类号 |
A61K31/69 |
代理机构 |
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