发明名称 PROCESS FOR THE PREPARATION OF ANHYDROUS ARIPIPRAZOLE CRYSTAL FORM II
摘要 The present invention relates to a process for preparation of aripiprazole crystal form II by recrystallizing aripiprazole in a mixture of acetone and 1-methoxy-2-propanol or a single solvent of 1-methoxy-2-propanol. The simple process according to the present invention can produce aripiprazole crystal form II with high purity and high yield in a mass scale.
申请公布号 WO2012134206(A3) 申请公布日期 2012.11.29
申请号 WO2012KR02349 申请日期 2012.03.30
申请人 DAEWOONG PHARMACEUTICAL CO., LTD.;CHOI, SOO JIN;OH, SEONG SOO;JIN, YONG SUK;KIM, YONG TAE;LEE, SEUNG JAE;SON, JEONG HYUN 发明人 CHOI, SOO JIN;OH, SEONG SOO;JIN, YONG SUK;KIM, YONG TAE;LEE, SEUNG JAE;SON, JEONG HYUN
分类号 C07D401/12;A61K31/4709;A61K31/496;A61P25/00 主分类号 C07D401/12
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