发明名称 A PROCESS FOR THE PREPARATION OF LASOFOXIFENE TARTRATE
摘要 <p>A solid crystalline form of 1-(2-[4-(6-methoxy-3,4-dihydronaphthalene-1-y) phenoxy]ethyl)pyrrolidine, and a preparing process thereof are provided. The aforesaid compound is a key intermediate in the synthesis of lasofoxifene. A process for preparing lasofoxifene, a process for purifying lasofoxifene tartrate, and a crystalline form of lasofoxifene tartrate are also provided.</p>
申请公布号 EP2424839(A4) 申请公布日期 2012.10.17
申请号 EP20100769411 申请日期 2010.04.27
申请人 GLENMARK GENERICS LIMITED 发明人 KHAN, MUBEEN AHMED;TRIVEDI, NIKHIL RASIKLAL;KANDASAMY, NAGAN NIRMALAN;PATIL, DAYAGHAN GANGADHAR;PANDEY, VIPIN KUMAR;SINHA, SUKUMAR
分类号 C07D207/08 主分类号 C07D207/08
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