发明名称 Novel Inhibitors
摘要 Novel heterocyclic derivatives of formula (I): or a pharmaceutically acceptable salt, solvate or polymorph thereof, including all tautomers and stereoisomers thereof, wherein Ra, n, R1 and R2 are as defined herein, as inhibitors of glutaminyl cyclase (QC, EC 2.3.2.5).
申请公布号 US2012237475(A1) 申请公布日期 2012.09.20
申请号 US201213422619 申请日期 2012.03.16
申请人 HEISER ULRICH;RAMSBECK DANIEL;PROBIODRUG AG 发明人 HEISER ULRICH;RAMSBECK DANIEL
分类号 A61K38/20;A61K31/4184;A61K31/4409;A61K31/454;A61K31/496;A61K31/5377;A61K31/541;A61K33/14;A61K38/10;A61K38/21;A61K39/395;A61P1/04;A61P1/18;A61P3/00;A61P5/00;A61P7/00;A61P9/00;A61P9/10;A61P15/08;A61P17/06;A61P19/02;A61P25/00;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P25/28;A61P29/00;A61P31/04;A61P35/00;A61P35/04;A61P37/00;A61P37/02;A61P37/06;C07D401/14;C07D403/10;C07D403/14;C07D405/14;C07D409/14;C07D413/14;C07D417/14 主分类号 A61K38/20
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