发明名称 |
SUBSTITUTED 2-ALKYL QUINAZOLINONE DERIVATIVES AS PARP INHIBITORS |
摘要 |
<p>The present invention provides compounds of formula (I), their use as PARP inhibitors as well as pharmaceutical compositions comprising said compounds of formula (I) wherein R1, R2, R3, L, X, Y and Z have defined meanings.</p> |
申请公布号 |
EP1763518(B1) |
申请公布日期 |
2012.01.11 |
申请号 |
EP20050756772 |
申请日期 |
2005.06.28 |
申请人 |
JANSSEN PHARMACEUTICA NV |
发明人 |
VAN DER AA, MARCEL JOZEF MARIA;VAN HEERTUM, ALBERTUS HENRICUS MARIA THERESIA;VAN DUN, JACOBUS ALPHONSUS JOSEPHUS;SOMERS, MARIA VICTORINA FRANCISCA;WOUTERS, WALTER BOUDEWIJN LEOPOLD |
分类号 |
C07D239/90;A61K31/517;A61P25/00;C07D239/91;C07D401/06;C07D401/12;C07D403/12;C07D405/12 |
主分类号 |
C07D239/90 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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