发明名称 CYCLOAMINO DERIVATIVES AS GPR119 ANTAGONISTS
摘要 <p>Therapeutic compounds are disclosed having the general formula (I) that are useful for the treatment of metabolic disorders, including type II diabetes. The compounds have activity as agonists of GPR119. Compounds having the stereochemistry of formula (la) may also demonstrate DPP-IV inhibitory activity.</p>
申请公布号 WO2011147951(A1) 申请公布日期 2011.12.01
申请号 WO2011EP58703 申请日期 2011.05.27
申请人 PROSIDION LIMITED;BARBA, OSCAR;BELL, JAMES, CHARLES;DUPREE, TOM, BANKSIA;FRY, PETER, TIMOTHY;BERTRAM, LISA, SARAH;FYFE, MATTHEW, COLIN, THOR;GATTRELL, WILLIAM;JEEVARATNAM, REVATHY, PERPETUA;KEILY, JOHN;KRULLE, THOMAS, MARTIN;MCDONALD, RUSSELL, WALKER;MORGAN, TREVOR;RASAMISON, CHRYSTELLE, MARIE;SCHOFIELD, KAREN, LESLEY;STEWART, ALAN, JOHN, WILLIAM;SWAIN, SIMON, ANDREW;WITHALL, DAVID, MATTHEW 发明人 BARBA, OSCAR;BELL, JAMES, CHARLES;DUPREE, TOM, BANKSIA;FRY, PETER, TIMOTHY;BERTRAM, LISA, SARAH;FYFE, MATTHEW, COLIN, THOR;GATTRELL, WILLIAM;JEEVARATNAM, REVATHY, PERPETUA;KEILY, JOHN;KRULLE, THOMAS, MARTIN;MCDONALD, RUSSELL, WALKER;MORGAN, TREVOR;RASAMISON, CHRYSTELLE, MARIE;SCHOFIELD, KAREN, LESLEY;STEWART, ALAN, JOHN, WILLIAM;SWAIN, SIMON, ANDREW;WITHALL, DAVID, MATTHEW
分类号 C07D401/14;A61K31/454;A61P3/10;C07D409/14;C07D413/14;C07D417/14;C07D487/04;C07D491/08 主分类号 C07D401/14
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