发明名称 |
PROCESS AND INTERMEDIATES FOR THE SYNTHESIS OF 8-[{1-(3,5-BIS-(TRIFLUOROMETHYL)PHENYL)-ETHOXY}-METHYL]-8-PHENYL-1,7-DIAZA-SPIRO[4.5]DECAN-2-ONE COMPOUNDS |
摘要 |
This application discloses a novel process to synthesize 8-[{1-(3,5-Bis-(trifluoromethyl)phenyl)-ethoxy}-methyl]-8-phenyl-1,7-diaza-spiro[4.5]decan-2-one compounds, which may be used, for example, as NK-1 inhibitor compounds in pharmaceutical preparations. |
申请公布号 |
KR20110067117(A) |
申请公布日期 |
2011.06.21 |
申请号 |
KR20117007788 |
申请日期 |
2009.09.04 |
申请人 |
OPKO HEALTH, INC. |
发明人 |
WU GEORGE G.;WERNE GERALD;FU XIAOYONG;ORR ROBERT K.;CHEN FRANK XING;CUI JIAN;SPRAGUE VICTORIA M.;ZHANG FUCHENG;XIE JI;ZENG LIANSHENG;CASTELLANOS LOUIS PETER;CHEN YUYIN;POIRIER MARC;MERGELSBERG INGRID |
分类号 |
C07D471/10;C07D207/26;C07D498/04 |
主分类号 |
C07D471/10 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|