发明名称 |
GLYCINE TRANSPORTER INHIBITORS |
摘要 |
<p>The present invention aims to provide novel compounds represented by formula [I] or pharmaceutically acceptable salts thereof: [Formula 1] which are useful for prevention or treatment of diseases such as schizophrenia, Alzheimer's disease, cognitive impairment, dementia, anxiety disorders (e.g., generalized anxiety disorder, panic disorder, obsessive-compulsive disorder, social anxiety disorder, post-traumatic stress disorder, specific phobias, acute stress disorder), depression, drug dependence, convulsion, tremor, pain, or sleep disorders, based on their inhibitory effect against glycine uptake.</p> |
申请公布号 |
WO2011007899(A1) |
申请公布日期 |
2011.01.20 |
申请号 |
WO2010JP62394 |
申请日期 |
2010.07.15 |
申请人 |
TAISHO PHARMACEUTICAL CO., LTD.;YASUHARA, AKITO;SAKAGAMI, KAZUNARI;OHTA, HIROSHI;HAYASHI, MASATO;SHIRASAKI, YOSHIHISA;YAMAMOTO, SHUJI;SHIMAZAKI, YOUICHI;ARAKI, YUKO;ABE, KUMI;SUN, XIANG-MIN |
发明人 |
YASUHARA, AKITO;SAKAGAMI, KAZUNARI;OHTA, HIROSHI;HAYASHI, MASATO;SHIRASAKI, YOSHIHISA;YAMAMOTO, SHUJI;SHIMAZAKI, YOUICHI;ARAKI, YUKO;ABE, KUMI;SUN, XIANG-MIN |
分类号 |
C07D233/90;A61K31/4164;A61K31/4196;A61P25/00;A61P25/04;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P43/00;C07D249/10 |
主分类号 |
C07D233/90 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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