CRYSTALLINE FORMS OF 4-[6-(6-METHANESULFONYL-2-METHYLPYRIDIN-3-YLAMINO)-5-METHOXY-PYRIMIDIN-4-YLOXY]-PIPERIDINE-1-CARBOXYLIC ACID ISOPROPYL ESTER
摘要
The present invention is directed to a novel crystalline forms of 4-[6-(6- methanesulfonyl-2-methyl-pyhdin-3-ylamino)-5-methoxy-pyhmidin-4-yloxy]- piperidine-1 -carboxylic acid isopropyl ester, pharmaceutical compositions containing said crystalline form and the use of said crystalline forms in the treatment of metabolic related disorders. The present invention is further directed to processes for the preparation of the crystalline forms of 4-[6-(6- methanesulfonyl-2-methyl-pyhdin-3-ylamino)-5-methoxy-pyhmidin-4-yloxy]- piperidine-1 -carboxylic acid isopropyl ester.
申请公布号
WO2010135505(A2)
申请公布日期
2010.11.25
申请号
WO2010US35536
申请日期
2010.05.20
申请人
JANSSEN PHARMACEUTICA NV;WELLS, KENNETH M.;FECH, GARY;WU, WENJU;FAWZY, NAGY E.
发明人
WELLS, KENNETH M.;FECH, GARY;WU, WENJU;FAWZY, NAGY E.