发明名称 |
Benzoxazepines as Inhibitors of PI3K/mTOR and Methods of Their Use and Manufacture |
摘要 |
The invention is directed to Compounds of Formula I: and pharmaceutically acceptable salts or solvates thereof, as well as methods of making and using the compounds.
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申请公布号 |
US2010298290(A1) |
申请公布日期 |
2010.11.25 |
申请号 |
US20100784254 |
申请日期 |
2010.05.20 |
申请人 |
EXELIXIS, INC. |
发明人 |
ANAND NEEL KUMAR;BLAZEY CHARLES M.;BOWLES OWEN JOSEPH;BUHR CHRIS ALLEN;BUSSENIUS JOERG;CURTIS JEFFRY KIMO;DEFINA STEVEN CHARLES;DUBENKO LARISA;HARRIS JASON R.;JACKSON-UGUETO EILEEN E.;JOSHI ANAGHA;KIM ANGIE INYOUNG;TSUHAKO AMY LEW;MA SUNGHOON;MANALO JEAN-CLAIRE LIMUN;NG STEPHANIE;PETO CSABA J.;RICE KENNETH D.;TSANG TSZE H.;ZAHARIA CRISTIANA A. |
分类号 |
A61K31/553;A61P35/00;A61P35/04;C07D413/14 |
主分类号 |
A61K31/553 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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