发明名称 Benzoxazepines as Inhibitors of PI3K/mTOR and Methods of Their Use and Manufacture
摘要 The invention is directed to Compounds of Formula I: and pharmaceutically acceptable salts or solvates thereof, as well as methods of making and using the compounds.
申请公布号 US2010298290(A1) 申请公布日期 2010.11.25
申请号 US20100784254 申请日期 2010.05.20
申请人 EXELIXIS, INC. 发明人 ANAND NEEL KUMAR;BLAZEY CHARLES M.;BOWLES OWEN JOSEPH;BUHR CHRIS ALLEN;BUSSENIUS JOERG;CURTIS JEFFRY KIMO;DEFINA STEVEN CHARLES;DUBENKO LARISA;HARRIS JASON R.;JACKSON-UGUETO EILEEN E.;JOSHI ANAGHA;KIM ANGIE INYOUNG;TSUHAKO AMY LEW;MA SUNGHOON;MANALO JEAN-CLAIRE LIMUN;NG STEPHANIE;PETO CSABA J.;RICE KENNETH D.;TSANG TSZE H.;ZAHARIA CRISTIANA A.
分类号 A61K31/553;A61P35/00;A61P35/04;C07D413/14 主分类号 A61K31/553
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