Processes for preparing 4-(phenoxy-5-methyl-pyrimidin-4-yloxy) piperidine-1-carboxylic acid derivatives and related compounds
摘要
Disclosed herein is a process for preparing an iodide salt compound of formula I, comprising of: reacting a compound of Formula II with a compound of Formula III in the presence of an iodide salt, wherein substituents are as defined within the specification. Also disclosed is a process for preparing a compound of Formula II by combining a compound of Formula IV with a compound of Formula V to form a mixture and then adding a base to said mixture to form a compound of Formula II.
申请公布号
NZ556218(A)
申请公布日期
2010.10.29
申请号
NZ20060556218
申请日期
2006.01.09
申请人
ARENA PHARMACEUTICALS, INC.
发明人
GHARBAOUI, TAWFIK;FRITCH, JOHN R;KRISHNAN, ASHWIN M;THROOP, BEVERLY WOLGAST;KATO, NAOMI S